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L-778123 hydrochloride

CAS No. 253863-00-2

L-778123 hydrochloride( L-778,123 hydrochloride )

Catalog No. M17457 CAS No. 253863-00-2

The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.

Purity : >98% (HPLC)

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HNMR

HPLC

MSDS

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2MG	34	In Stock
5MG	55	In Stock
10MG	80	In Stock
25MG	143	In Stock
50MG	236	In Stock
100MG	398	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

L-778123 hydrochloride
Note

Research use only, not for human use.
Brief Description

The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.
Description

The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.
In Vitro

——
In Vivo

——
Synonyms

L-778,123 hydrochloride
Pathway

Endocrinology/Hormones
Target

Estrogen Receptor/ERR
Recptor

Farnesyl transferase (FTase)
Research Area

Cancer
Indication

——

Chemical Information

CAS Number

253863-00-2
Formula Weight

442.34
Molecular Formula

C22H21Cl2N5O
Purity

>98% (HPLC)
Solubility

DMSO : ≥ 25 mg/mL; 56.52 mM
SMILES

c1cc(cc(c1)N1CCN(Cc2cncn2Cc2ccc(cc2)C#N)CC1=O)Cl.Cl
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Lobell RB, et al. Mol Y Ther. 2002 Jul;1(9):747-58.

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